HCAR2 (hydroxycarboxylic acid receptor 2)

2011-10-01  

Identity

HGNC
LOCATION
12q24.31
LOCUSID
ALIAS
GPR109A,HCA2,HM74a,HM74b,NIACR1,PUMAG,Puma-g

Other Information

Locus ID:

NCBI: 338442
MIM: 609163
HGNC: 24827
Ensembl: ENSG00000182782

Variants:

dbSNP: 338442
ClinVar: 338442
TCGA: ENSG00000182782
COSMIC: HCAR2

RNA/Proteins

Gene IDTranscript IDUniprot
ENSG00000182782ENST00000328880Q8TDS4
ENSG00000182782ENST00000328880A0A4Y1JWQ0

Expression (GTEx)

0
10
20
30
40
50
60
70
80

Pathways

PathwaySourceExternal ID
cAMP signaling pathwayKEGGhsa04024
cAMP signaling pathwayKEGGko04024
Signal TransductionREACTOMER-HSA-162582
Signaling by GPCRREACTOMER-HSA-372790
GPCR ligand bindingREACTOMER-HSA-500792
Class A/1 (Rhodopsin-like receptors)REACTOMER-HSA-373076
Hydroxycarboxylic acid-binding receptorsREACTOMER-HSA-3296197
GPCR downstream signalingREACTOMER-HSA-388396
G alpha (i) signalling eventsREACTOMER-HSA-418594

Protein levels (Protein atlas)

Not detected
Low
Medium
High

PharmGKB

Entity IDNameTypeEvidenceAssociationPKPDPMIDs
PA450617niacinChemicalVariantAnnotationnot associatedPD

References

Pubmed IDYearTitleCitations
375780112023Ebola Virus Infection Induces HCAR2 Expression Leading to Cell Death.0
379322632023Structural basis for ligand recognition and signaling of hydroxy-carboxylic acid receptor 2.3
379336502023[GPR109A partly mediates inhibitory effects of β-hydroxybutyric acid on lung adenocarcinoma cell proliferation, migration and invasion].0
380075722023Parabacteroides distasonis ameliorates insulin resistance via activation of intestinal GPR109a.3
375780112023Ebola Virus Infection Induces HCAR2 Expression Leading to Cell Death.0
379322632023Structural basis for ligand recognition and signaling of hydroxy-carboxylic acid receptor 2.3
379336502023[GPR109A partly mediates inhibitory effects of β-hydroxybutyric acid on lung adenocarcinoma cell proliferation, migration and invasion].0
380075722023Parabacteroides distasonis ameliorates insulin resistance via activation of intestinal GPR109a.3
347773632021GPR Expression in Intestinal Biopsies From SCT Patients Is Upregulated in GvHD and Is Suppressed by Broad-Spectrum Antibiotics.6
348528022021Rare and potentially pathogenic variants in hydroxycarboxylic acid receptor genes identified in breast cancer cases.2
347773632021GPR Expression in Intestinal Biopsies From SCT Patients Is Upregulated in GvHD and Is Suppressed by Broad-Spectrum Antibiotics.6
348528022021Rare and potentially pathogenic variants in hydroxycarboxylic acid receptor genes identified in breast cancer cases.2
317343542020Clostridium butyricum, a butyrate-producing probiotic, inhibits intestinal tumor development through modulating Wnt signaling and gut microbiota.176
318581052020Niacin Ameliorates Hepatic Steatosis by Inhibiting De Novo Lipogenesis Via a GPR109A-Mediated PKC-ERK1/2-AMPK Signaling Pathway in C57BL/6 Mice Fed a High-Fat Diet.16
317343542020Clostridium butyricum, a butyrate-producing probiotic, inhibits intestinal tumor development through modulating Wnt signaling and gut microbiota.176

Citation

Dessen P

HCAR2 (hydroxycarboxylic acid receptor 2)

Atlas Genet Cytogenet Oncol Haematol. 2011-10-01

Online version: http://atlasgeneticsoncology.org/gene/52400/hcar2