GRK3 (G protein-coupled receptor kinase 3)

2006-10-01  

Identity

HGNC
LOCATION
22q12.1
LOCUSID
ALIAS
ADRBK2,BARK2
FUSION GENES

Other Information

Locus ID:

NCBI: 157
MIM: 109636
HGNC: 290
Ensembl: ENSG00000100077

Variants:

dbSNP: 157
ClinVar: 157
TCGA: ENSG00000100077
COSMIC: GRK3

RNA/Proteins

Gene IDTranscript IDUniprot
ENSG00000100077ENST00000324198P35626
ENSG00000100077ENST00000324198A0A024R1D8
ENSG00000100077ENST00000455558H7C099
ENSG00000100077ENST00000619906Q8N433

Expression (GTEx)

0
5
10
15
20
25
30
35

Pathways

PathwaySourceExternal ID
Hedgehog signaling pathwayKEGGko04340
Olfactory transductionKEGGko04740
Hedgehog signaling pathwayKEGGhsa04340
Olfactory transductionKEGGhsa04740
Chemokine signaling pathwayKEGGko04062
Chemokine signaling pathwayKEGGhsa04062
EndocytosisKEGGko04144
EndocytosisKEGGhsa04144
Glutamatergic synapseKEGGko04724
Glutamatergic synapseKEGGhsa04724
Morphine addictionKEGGhsa05032
Morphine addictionKEGGko05032
Signal TransductionREACTOMER-HSA-162582
Signaling by GPCRREACTOMER-HSA-372790
GPCR downstream signalingREACTOMER-HSA-388396
G alpha (s) signalling eventsREACTOMER-HSA-418555
Vesicle-mediated transportREACTOMER-HSA-5653656
Membrane TraffickingREACTOMER-HSA-199991
Clathrin-mediated endocytosisREACTOMER-HSA-8856828
Cargo recognition for clathrin-mediated endocytosisREACTOMER-HSA-8856825

Protein levels (Protein atlas)

Not detected
Low
Medium
High

PharmGKB

Entity IDNameTypeEvidenceAssociationPKPDPMIDs
PA30616MAPK1GenePathwayassociated
PA39ADRB2GenePathwayassociated
PA62ATP1A1GenePathwayassociated23788015

References

Pubmed IDYearTitleCitations
369071392023TEAD3 inhibits the proliferation and metastasis of prostate cancer via suppressing ADRBK2.1
370480542023Aged G Protein-Coupled Receptor Kinase 3 (Grk3)-Deficient Mice Exhibit Enhanced Osteoclastogenesis and Develop Bone Lesions Analogous to Human Paget's Disease of Bone.0
375432782023A novel GRK3-HDAC2 regulatory pathway is a key direct link between neuroendocrine differentiation and angiogenesis in prostate cancer progression.1
369071392023TEAD3 inhibits the proliferation and metastasis of prostate cancer via suppressing ADRBK2.1
370480542023Aged G Protein-Coupled Receptor Kinase 3 (Grk3)-Deficient Mice Exhibit Enhanced Osteoclastogenesis and Develop Bone Lesions Analogous to Human Paget's Disease of Bone.0
375432782023A novel GRK3-HDAC2 regulatory pathway is a key direct link between neuroendocrine differentiation and angiogenesis in prostate cancer progression.1
330606472020Dissecting the roles of GRK2 and GRK3 in μ-opioid receptor internalization and β-arrestin2 recruitment using CRISPR/Cas9-edited HEK293 cells.18
330606472020Dissecting the roles of GRK2 and GRK3 in μ-opioid receptor internalization and β-arrestin2 recruitment using CRISPR/Cas9-edited HEK293 cells.18
316045292019The N-termini of GRK2 and GRK3 simulate the stimulating effects of RKIP on β-adrenoceptors.4
316045292019The N-termini of GRK2 and GRK3 simulate the stimulating effects of RKIP on β-adrenoceptors.4
292547922018High expression of GRK3 is associated with favorable prognosis in pancreatic ductal adenocarcinoma.5
292547922018High expression of GRK3 is associated with favorable prognosis in pancreatic ductal adenocarcinoma.5
294452492017Overexpression of GRK3, Promoting Tumor Proliferation, Is Predictive of Poor Prognosis in Colon Cancer.8
294452492017Overexpression of GRK3, Promoting Tumor Proliferation, Is Predictive of Poor Prognosis in Colon Cancer.8
270497552016G Protein Coupled Receptor Kinase 3 Regulates Breast Cancer Migration, Invasion, and Metastasis.29

Citation

Dessen P

GRK3 (G protein-coupled receptor kinase 3)

Atlas Genet Cytogenet Oncol Haematol. 2006-10-01

Online version: http://atlasgeneticsoncology.org/gene/43107/gene-fusions-explorer/meetings/