AKR1C4 (aldo-keto reductase family 1 member C4)

2017-04-01  

Identity

HGNC
LOCATION
10p15.1
LOCUSID
ALIAS
3-alpha-HSD,C11,CDR,CHDR,DD-4,DD4,HAKRA
FUSION GENES

Other Information

Locus ID:

NCBI: 1109
MIM: 600451
HGNC: 387
Ensembl: ENSG00000198610

Variants:

dbSNP: 1109
ClinVar: 1109
TCGA: ENSG00000198610
COSMIC: AKR1C4

RNA/Proteins

Gene IDTranscript IDUniprot
ENSG00000198610ENST00000263126P17516
ENSG00000198610ENST00000380448P17516

Expression (GTEx)

0
50
100
150
200

Pathways

PathwaySourceExternal ID
Primary bile acid biosynthesisKEGGko00120
Steroid hormone biosynthesisKEGGko00140
Primary bile acid biosynthesisKEGGhsa00120
Steroid hormone biosynthesisKEGGhsa00140
Metabolic pathwaysKEGGhsa01100
Bile acid biosynthesis, cholesterol => cholate/chenodeoxycholateKEGGhsa_M00104
Bile acid biosynthesis, cholesterol => cholate/chenodeoxycholateKEGGM00104
Signal TransductionREACTOMER-HSA-162582
Visual phototransductionREACTOMER-HSA-2187338
Retinoid metabolism and transportREACTOMER-HSA-975634
MetabolismREACTOMER-HSA-1430728
Metabolism of lipids and lipoproteinsREACTOMER-HSA-556833
Bile acid and bile salt metabolismREACTOMER-HSA-194068
Synthesis of bile acids and bile saltsREACTOMER-HSA-192105
Synthesis of bile acids and bile salts via 7alpha-hydroxycholesterolREACTOMER-HSA-193368
Synthesis of bile acids and bile salts via 24-hydroxycholesterolREACTOMER-HSA-193775
Synthesis of bile acids and bile salts via 27-hydroxycholesterolREACTOMER-HSA-193807
Metabolism of vitamins and cofactorsREACTOMER-HSA-196854
Metabolism of fat-soluble vitaminsREACTOMER-HSA-6806667

Protein levels (Protein atlas)

Not detected
Low
Medium
High

PharmGKB

Entity IDNameTypeEvidenceAssociationPKPDPMIDs
PA449212daunorubicinChemicalVariantAnnotationassociatedPK20837989
PA449563exemestaneChemicalClinicalAnnotationassociatedPK27111237

References

Pubmed IDYearTitleCitations
282599892017Mefenamic acid enhances anticancer drug sensitivity via inhibition of aldo-keto reductase 1C enzyme activity.20
282599892017Mefenamic acid enhances anticancer drug sensitivity via inhibition of aldo-keto reductase 1C enzyme activity.20
241891852014Role of aldo-keto reductase family 1 (AKR1) enzymes in human steroid metabolism.80
241891852014Role of aldo-keto reductase family 1 (AKR1) enzymes in human steroid metabolism.80
223568242012Polymorphisms in AKR1C4 and HSD3B2 and differences in serum DHEAS and progesterone are associated with paranoid ideation during mania or hypomania in bipolar disorder.12
223568242012Polymorphisms in AKR1C4 and HSD3B2 and differences in serum DHEAS and progesterone are associated with paranoid ideation during mania or hypomania in bipolar disorder.12
215211742011Stereospecific reduction of 5β-reduced steroids by human ketosteroid reductases of the AKR (aldo-keto reductase) superfamily: role of AKR1C1-AKR1C4 in the metabolism of testosterone and progesterone via the 5β-reductase pathway.21
215701272011AKR1C4 gene variant associated with low euthymic serum progesterone and a history of mood irritability in males with bipolar disorder.7
215211742011Stereospecific reduction of 5β-reduced steroids by human ketosteroid reductases of the AKR (aldo-keto reductase) superfamily: role of AKR1C1-AKR1C4 in the metabolism of testosterone and progesterone via the 5β-reductase pathway.21
215701272011AKR1C4 gene variant associated with low euthymic serum progesterone and a history of mood irritability in males with bipolar disorder.7
196921682010Genetic susceptibility to distinct bladder cancer subphenotypes.30
202019262010Human variation in alcohol response is influenced by variation in neuronal signaling genes.52
202148022010Genetic variation in the estrogen metabolic pathway and mammographic density as an intermediate phenotype of breast cancer.11
196921682010Genetic susceptibility to distinct bladder cancer subphenotypes.30
202019262010Human variation in alcohol response is influenced by variation in neuronal signaling genes.52

Citation

Dessen P

AKR1C4 (aldo-keto reductase family 1 member C4)

Atlas Genet Cytogenet Oncol Haematol. 2017-04-01

Online version: http://atlasgeneticsoncology.org/gene/56854/gene-fusions/meetings/